Sfoglia per Autore
Drug–Drug Interaction Studies of Esmethadone (REL-1017) Involving CYP3A4- and CYP2D6-Mediated Metabolism
2023 Ferri, N.; De Martin, S.; Stuart, J.; Traversa, S.; Folli, F.; Pappagallo, M.; O’Gorman, C.; Guidetti, C.; Mattarei, A.; Inturrisi, C. E.; Manfredi, P. L.
Toward a New Era in the Management of Hepatocellular Carcinoma: Novel Perspectives on Therapeutic Options and Biomarkers
2023 Gabbia, Daniela; De Martin, Sara
Tumor Mutational Burden for Predicting Prognosis and Therapy Outcome of Hepatocellular Carcinoma
2023 Gabbia, Daniela; De Martin, Sara
Esmethadone-HCl (REL-1017): a promising rapid antidepressant
2023 Fava, Maurizio; Stahl, Stephen M; De Martin, Sara; Mattarei, Andrea; Bettini, Ezio; Comai, Stefano; Alimonti, Andrea; Bifari, Francesco; Pani, Luca; Folli, Franco; Guidetti, Clotilde; Furlan, Alberto; Sgrignani, Jacopo; Locatelli, Patrizia; Cavalli, Andrea; O'Gorman, Cedric; Traversa, Sergio; Inturrisi, Charles E; Pappagallo, Marco; Manfredi, Paolo L
The novel uncompetitive NMDA receptor antagonist esmethadone (REL-1017) has no meaningful abuse potential in recreational drug users
2023 Shram, Megan J; Henningfield, Jack E; Apseloff, Glen; Gorodetzky, Charles W; De Martin, Sara; Vocci, Frank L; Sapienza, Frank L; Kosten, Thomas R; Huston, Jeff; Buchhalter, August; Ashworth, Judy; Lanier, Ryan; Folli, Franco; Mattarei, Andrea; Guidetti, Clotilde; Comai, Stefano; O'Gorman, Cedric; Traversa, Sergio; Inturrisi, Charles E; Manfredi, Paolo L; Pappagallo, Marco
The phenolic compounds tyrosol and hydroxytyrosol counteract liver fibrogenesis via the transcriptional modulation of NADPH oxidases and oxidative stress-related miRNAs
2023 Gabbia, Daniela; Carpi, Sara; Sarcognato, Samantha; Zanotto, Ilaria; Sayaf, Katia; Colognesi, Martina; Polini, Beatrice; Digiacomo, Maria; Macchia, Marco; Nieri, Paola; Carrara, Maria; Cazzagon, Nora; Russo, Francesco Paolo; Guido, Maria; De Martin, Sara
Subanalysis of Subjective Cognitive Measures From a Phase 2, Double-Blind, Randomized Trial of REL-1017 in Patients With Major Depressive Disorder
2023 Guidetti, Clotilde; Serra, Giulia; Pani, Luca; Pappagallo, Marco; Maglio, Gino; Martin, Sara De; Mattarei, Andrea; Folli, Franco; Manfredi, Paolo L; Fava, Maurizio
Sex Drives Functional Changes in the Progression and Regression of Liver Fibrosis
2023 Sayaf, K.; Zanotto, I.; Gabbia, D.; Alberti, D.; Pasqual, G.; Zaramella, A.; Fantin, A.; De Martin, S.; Russo, F. P.
Anti-HER2 Super Stealth Immunoliposomes for Targeted-Chemotherapy
2023 Canato, Elena; Grigoletto, Antonella; Zanotto, Ilaria; Tedeschini, Tommaso; Campara, Benedetta; Quaglio, Giovanna; Toffoli, Giuseppe; Mandracchia, Delia; Dinarello, Alberto; Tiso, Natascia; Argenton, Francesco; Sayaf, Katia; Guido, Maria; Gabbia, Daniela; De Martin, Sara; Pasut, Gianfranco
Update on the Pharmacological Treatment of Primary Biliary Cholangitis
2022 Floreani, A; Gabbia, D; De Martin, S
A Nutraceutical Formulation Containing Brown Algae Reduces Hepatic Lipid Accumulation by Modulating Lipid Metabolism and Inflammation in Experimental Models of NAFLD and NASH
2022 Gabbia, Daniela; Roverso, Marco; Zanotto, Ilaria; Colognesi, Martina; Sayaf, Katia; Sarcognato, Samantha; Arcidiacono, Diletta; Zaramella, Alice; Realdon, Stefano; Ferri, Nicola; Guido, Maria; Russo, Francesco Paolo; Bogialli, Sara; Carrara, Maria; De Martin, Sara
REL-1017 (Esmethadone) May Rapidly Reduce Dissociative Symptoms in Adults With Major Depressive Disorder Unresponsive to Standard Antidepressants: A Report of 2 Cases
2022 Guidetti, Clotilde; Serra, Giulia; Pani, Luca; Pappagallo, Marco; Maglio, Gino; Trasolini, Monia; De Martin, Sara; Mattarei, Andrea; Bifari, Francesco; Folli, Franco; Manfredi, Paolo L; Fava, Maurizio
PCSK9 promotes arterial medial calcification
2022 Lupo, M. G.; Bressan, A.; Donato, M.; Canzano, P.; Camera, M.; Poggio, P.; Greco, M. F.; Garofalo, M.; De Martin, S.; Panighel, G.; Ruscica, M.; Baragetti, A.; Bollati, V.; Faggin, E.; Rattazzi, M.; Catapano, A. L.; Ferri, N.
The N-Methyl-D-Aspartate Receptor Blocker REL-1017 (Esmethadone) Reduces Calcium Influx Induced by Glutamate, Quinolinic Acid, and Gentamicin
2022 Bettini, Ezio; De Martin, Sara; Mattarei, Andrea; Pappagallo, Marco; Stahl, Stephen M; Bifari, Francesco; Inturrisi, Charles E; Folli, Franco; Traversa, Sergio; Manfredi, Paolo L
Primary biliary cholangitis: Perception and expectation of illness in Italian patients
2022 Floreani, A.; Scaffidi, M.; Coco, B.; Giannini, E. G.; Labanca, S.; Bonaiuto, E.; De Martin, S.; Invernizzi, P.; Carbone, M.; Alvaro, D.; Bragazzi, M. C.; Calvaruso, V.; Cossiga, V.; Cazzagon, N.
The nuclear receptor PXR in chronic liver disease
2022 Sayaf, K.; Zanotto, I.; Russo, F. P.; Gabbia, D.; De Martin, S.
Pharmacological Comparative Characterization of REL-1017 (Esmethadone-HCl) and Other NMDAR Channel Blockers in Human Heterodimeric N-Methyl-D-Aspartate Receptors
2022 Bettini, Ezio; Stahl, Stephen M; De Martin, Sara; Mattarei, Andrea; Sgrignani, Jacopo; Carignani, Corrado; Nola, Selena; Locatelli, Patrizia; Pappagallo, Marco; Inturrisi, Charles E; Bifari, Francesco; Cavalli, Andrea; Alimonti, Andrea; Pani, Luca; Fava, Maurizio; Traversa, Sergio; Folli, Franco; Manfredi, Paolo L
Esmethadone (REL-1017) and Other Uncompetitive NMDAR Channel Blockers May Improve Mood Disorders via Modulation of Synaptic Kinase-Mediated Signaling
2022 Stahl, Stephen M; De Martin, Sara; Mattarei, Andrea; Bettini, Ezio; Pani, Luca; Guidetti, Clotilde; Folli, Franco; de Somer, Marc; Traversa, Sergio; Inturrisi, Charles E; Pappagallo, Marco; Gentilucci, Marco; Alimonti, Andrea; Fava, Maurizio; Manfredi, Paolo L
COVID-19 and Autoimmune Liver Diseases
2022 Floreani, Annarosa; De Martin, Sara
Self-Emulsifying Formulations to Increase the Oral Bioavailability of 4,6,4′-Trimethylangelicin as a Possible Treatment for Cystic Fibrosis
2022 Franceschinis, Erica; Roverso, Marco; Gabbia, Daniela; De Martin, Sara; Brusegan, Matteo; Vaccarin, Christian; Bogialli, Sara; Chilin, Adriana
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