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Mostrati risultati da 1 a 20 di 34
Titolo Data di pubblicazione Autori Rivista Serie Titolo libro
New bioisosteric sulphur-containing choline kinase inhibitors with a tracked mode of action 2023 Mariotto, ElenaMarchioro, ChiaraViola, Giampietro + EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - -
Molecular and functional profiling of chemotolerant cells unveils nucleoside metabolism-dependent vulnerabilities in medulloblastoma 2023 Mariotto, ElenaRampazzo, ElenaBortolozzi, RobertaRruga, FatlumManfreda, LorenzoMarchioro, ChiaraCanton, MartinaBresolin, SilviaViola, GiampietroPersano, Luca + ACTA NEUROPATHOLOGICA COMMUNICATIONS - -
Design, synthesis and biological evaluation of novel 2,4-thiazolidinedione derivatives able to target the human BAG3 protein 2023 Marchioro, ChiaraCanton, MartinaFavaro, AnnagiuliaSturlese, MattiaViola, GiampietroMariotto, Elena + EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - -
Identification of Homoharringtonine as a potent inhibitor of glioblastoma cell proliferation and migration 2023 Maule, FrancescaManfreda, LorenzoMariotto, ElenaBresolin, SilviaCani, AliceBortolozzi, RobertaCorallo, DianaViola, GiampietroRampazzo, ElenaPersano, Luca + TRANSLATIONAL RESEARCH - -
New bioisosteric sulphur-containing choline kinase inhibitors with a tracked mode of action 2023 Mariotto, ElenaMarchioro, ChiaraViola, Giampietro + EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - -
Design, Synthesis and Biological Investigation of 2-Anilino Triazolopyrimidines as Tubulin Polymerization Inhibitors with Anticancer Activities 2022 Corallo, DianaAveic, SanjaManfreda, LorenzoMariotto, ElenaViola, Giampietro + PHARMACEUTICALS - -
Histone Deacetylase Inhibitors Impair Glioblastoma Cell Motility and Proliferation 2022 Rampazzo E.Manfreda L.Bresolin S.Cani A.Mariotto E.Bortolozzi R.Viola G.Persano L. + CANCERS - -
Cinnamic acid derivatives linked to arylpiperazines as novel potent inhibitors of tyrosinase activity and melanin synthesis 2022 Corallo D.Aveic S.Mariotto E.Viola G.Bortolozzi R. + EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - -
Design, Synthesis and Biological Investigation of 2-Anilino Triazolopyrimidines as Tubulin Polymerization Inhibitors with Anticancer Activities 2022 Corallo, DianaAveic, SanjaManfreda, LorenzoMariotto, ElenaBortolozzi, RobertaViola, Giampietro + PHARMACEUTICALS - -
Biological Evaluation of New Thienopyridinium and Thienopyrimidinium Derivatives as Human Choline Kinase Inhibitors 2022 Mariotto E.Viola G. + PHARMACEUTICS - -
Synthesis and Biological Evaluation of Highly Active 7-Anilino Triazolopyrimidines as Potent Antimicrotubule Agents 2022 Corallo, DianaAveic, SanjaMilan, NoemiMariotto, ElenaViola, GiampietroBortolozzi, Roberta + PHARMACEUTICS - -
Anticancer and structure activity relationship of non-symmetrical choline kinase inhibitors 2021 Mariotto E.Viola G. + PHARMACEUTICS - -
A facile synthesis of diaryl pyrroles led to the discovery of potent colchicine site antimitotic agents 2021 Rruga F.Mariotto E.Viola G.Bortolozzi R. + EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - -
BAG1 down-regulation increases chemo-sensitivity of acute lymphoblastic leukaemia cells 2021 Mariotto E.Corallo D.Giarin E.Pigazzi M.Basso G.Viola G.Aveic S. + JOURNAL OF CELLULAR AND MOLECULAR MEDICINE - -
Developing novel classes of protein kinase CK1δ inhibitors by fusing [1,2,4]triazole with different bicyclic heteroaromatic systems 2021 Bissaro M.Mariotto E.Bortolozzi R.Viola G.Cozza G.Moro S. + EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - -
Autophagic flux inhibition enhances cytotoxicity of the receptor tyrosine kinase inhibitor ponatinib 2020 Corallo, DianaMariotto, ElenaCaicci, FedericoViola, GiampietroAveic, Sanja + JOURNAL OF EXPERIMENTAL & CLINICAL CANCER RESEARCH - -
A BAG's life: Every connection matters in cancer 2020 Mariotto E.Viola G.Aveic S. + PHARMACOLOGY & THERAPEUTICS - -
Synthesis, biological evaluation, in silico modeling and crystallization of novel small monocationic molecules with potent antiproliferative activity by dual mechanism 2020 Mariotto E.Viola G. + EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - -
Design, synthesis, in vitro and in vivo biological evaluation of 2-amino-3-aroylbenzo[b]furan derivatives as highly potent tubulin polymerization inhibitors 2020 Rruga, FatlumMariotto, ElenaViola, GiampietroBortolozzi, Roberta + EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - -
Potent In Vitro and In Vivo Anticancer Activity of New Bipyridine and Bipyrimidine Gold (III) Dithiocarbamate Derivatives 2019 Mariotto, Elena + CANCERS - -
Mostrati risultati da 1 a 20 di 34
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