Sfoglia per Autore
Stereocontrolled access to thioisosteres of nucleoside di- and triphosphates
2024 Zhang, Hai-Jun; Ociepa, Michał; Nassir, Molhm; Zheng, Bin; Lewicki, Sarah A.; Salmaso, Veronica; Baburi, Helay; Nagel, Jessica; Mirza, Salahuddin; Bueschbell, Beatriz; Al-Hroub, Haneen; Perzanowska, Olga; Lin, Ziqin; Schmidt, Michael A.; Eastgate, Martin D.; Jacobson, Kenneth A.; Müller, Christa E.; Kowalska, Joanna; Jemielity, Jacek; Baran, Phil S.
Fluorescent A2A and A3 adenosine receptor antagonists as flow cytometry probes
2023 Toti, Kiran S; Campbell, Ryan G; Lee, Hobin; Salmaso, Veronica; Suresh, R Rama; Gao, Zhan-Guo; Jacobson, Kenneth A
Thermal Titration Molecular Dynamics (TTMD): Not Your Usual Post-Docking Refinement
2023 Menin, Silvia; Pavan, Matteo; Salmaso, Veronica; Sturlese, Mattia; Moro, Stefano
Pyrazolo-triazolo-pyrimidine Scaffold as a Molecular Passepartout for the Pan-Recognition of Human Adenosine Receptors
2023 Salmaso, Veronica; Persico, Margherita; Da Ros, Tatiana; Spalluto, Giampiero; Kachler, Sonja; Klotz, Karl-Norbert; Moro, Stefano; Federico, Stephanie
First Potent Macrocyclic A3 Adenosine Receptor Agonists Reveal G-Protein and β-Arrestin2 Signaling Preferences
2023 Tosh, Dilip K.; Fisher, Courtney L.; Salmaso, Veronica; Wan, Tina C.; Campbell, Ryan G.; Chen, Eric; Gao, Zhan-Guo; Auchampach, John A.; Jacobson, Kenneth A.
Thermal titration molecular dynamics (TTMD): shedding light on the stability of RNA-small molecule complexes
2023 Dodaro, Andrea; Pavan, Matteo; Menin, Silvia; Salmaso, Veronica; Sturlese, Mattia; Moro, Stefano
[1,2,4]Triazolo[1,5‐c]pyrimidines as Tools to Investigate A3 Adenosine Receptors in Cancer Cell Lines
2023 Federico, Stephanie; Persico, Margherita; Trevisan, Letizia; Biasinutto, Chiara; Bolcato, Giovanni; Salmaso, Veronica; Da Ros, Tatiana; Gianferrara, Teresa; Prencipe, Filippo; Kachler, Sonja; Klotz, Karl‐norbert; Pacor, Sabrina; Moro, Stefano; Spalluto, Giampiero
2-Amino-5-arylethynyl-thiophen-3-yl-(phenyl)methanones as A1 Adenosine Receptor Positive Allosteric Modulators
2023 Oliva, Paola; Suresh, R. Rama; Pasquini, Silvia; Salmaso, Veronica; Will, Edward J.; Tosh, Dilip K.; Gao, Zhan-Guo; Liu, Naili; Gavrilova, Oksana; Vincenzi, Fabrizio; Varani, Katia; Jacobson, Kenneth A.
Structure-Activity Relationship of 3-Methylcytidine-5'-α,β-methylenediphosphates as CD73 Inhibitors
2022 Scortichini, Mirko; Idris, Riham Mohammed; Moschütz, Susanne; Keim, Antje; Salmaso, Veronica; Dobelmann, Clemens; Oliva, Paola; Losenkova, Karolina; Irjala, Heikki; Vaittinen, Samuli; Sandholm, Jouko; Yegutkin, Gennady G; Sträter, Norbert; Junker, Anna; Müller, Christa E; Jacobson, Kenneth A
Selective A3 Adenosine Receptor Antagonist Radioligand for Human and Rodent Species
2022 Suresh, R Rama; Gao, Zhan-Guo; Salmaso, Veronica; Chen, Eric; Campbell, Ryan G; Poe, Russell B; Liston, Theodore E; Jacobson, Kenneth A
Bridged Piperidine Analogues of a High Affinity Naphthalene-Based P2Y14R Antagonist
2022 Wen, Zhiwei; Salmaso, Veronica; Jung, Young-Hwan; Phung, Ngan B; Gopinatth, Varun; Shah, Qasim; Patterson, Alexandra T; Randle, John C R; Chen, Zhoumou; Salvemini, Daniela; Lieberman, David I; Whitehead, Gregory S; Karcz, Tadeusz P; Cook, Donald N; Jacobson, Kenneth A
Synthesis and Effect of Conformationally Locked Carbocyclic Guanine Nucleotides on Dynamin
2022 Toti, Kiran S; Jimah, John R; Salmaso, Veronica; Hinshaw, Jenny E; Jacobson, Kenneth A
A3 adenosine receptor agonists containing dopamine moieties for enhanced interspecies affinity
2022 Tosh, Dilip K; Salmaso, Veronica; Campbell, Ryan G; Rao, Harsha; Bitant, Amelia; Pottie, Eline; Stove, Christophe P; Liu, Naili; Gavrilova, Oksana; Gao, Zhan-Guo; Auchampach, John A; Jacobson, Kenneth A
Structure-Activity Studies of 1H-Imidazo[4,5-c]quinolin-4-amine Derivatives as A3 Adenosine Receptor Positive Allosteric Modulators
2022 Fallot, Lucas B; Suresh, R Rama; Fisher, Courtney L; Salmaso, Veronica; O'Connor, Robert D; Kaufman, Noy; Gao, Zhan-Guo; Auchampach, John A; Jacobson, Kenneth A
Purinergic GPCR transmembrane residues involved in ligand recognition and dimerization
2021 Salmaso, V.; Jain, S.; Jacobson, K. A.
Expanding the repertoire of methanocarba nucleosides from purinergic signaling to diverse targets
2021 Jacobson, Kenneth A; Salmaso, Veronica; Suresh, R Rama; Tosh, Dilip K
Structure-Activity Relationship of Heterocyclic P2Y14Receptor Antagonists: Removal of the Zwitterionic Character with Piperidine Bioisosteres
2021 Jung, Y. -H.; Salmaso, V.; Wen, Z.; Bennett, J. M.; Phung, N. B.; Lieberman, D. I.; Gopinatth, V.; Randle, J. C. R.; Chen, Z.; Salvemini, D.; Karcz, T. P.; Cook, D. N.; Jacobson, K. A.
Amphiphilic peptide-based MMP3 inhibitors for intra-articular treatment of knee OA
2021 Guarise, C.; Ceradini, D.; Tessari, M.; Pavan, M.; Moro, S.; Salmaso, V.; Barbera, C.; Beninatto, R.; Galesso, D.
Truncated (N)-Methanocarba Nucleosides as Partial Agonists at Mouse and Human A3 Adenosine Receptors: Affinity Enhancement by N6-(2-Phenylethyl) Substitution
2020 Tosh, D. K.; Salmaso, V.; Rao, H.; Bitant, A.; Fisher, C. L.; Lieberman, D. I.; Vorbruggen, H.; Reitman, M. L.; Gavrilova, O.; Gao, Z. -G.; Auchampach, J. A.; Jacobson, K. A.
Survey of ribose ring pucker of signaling nucleosides and nucleotides
2020 Salmaso, V.; Jacobson, K. A.
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