Sfoglia per Autore
Synthesis, structural and computational study, DNA binding and cytotoxic activity of Cu(II) complexes of 6- and 7-chloro-2-oxo-1,2-dihydroquinoline-3-carbaldehyde-2-furoyl-hydrazones
2024 Thirunavukkarasu, Thangavel; Sparkes, Hazel A.; Gandin, Valentina; Marzano, Cristina; Bertani, Roberta; Mozzon, Mirto; Scettri, Anna; Albinati, Alberto; Demartin, Francesco; Casella, Girolamo; Ferrante, Francesco; Zoleo, Alfonso; Sgarbossa, Paolo; Natarajan, Karuppannan
Novel design of dual-action Pt(iv) anticancer pro-drugs based on cisplatin and derivatives of the tyrosine kinase inhibitors imatinib and nilotinib
2023 Beirne, Darren Fergal; Farkaš, Barbara; Donati, Chiara; Gandin, Valentina; Rozas, Isabel; Velasco-Torrijos, Trinidad; Montagner, Diego
Oral Anticancer Heterobimetallic PtIV−AuIComplexes Show High In Vivo Activity and Low Toxicity
2023 Babu, Tomer; Ghareeb, Hiba; Basu, Uttara; Schueffl, Hemma; Theiner, Sarah; Heffeter, Petra; Koellensperger, Gunda; Metanis, Norman; Gandin, Valentina; Ott, Ingo; Schmidt, Claudia; Gibson, Dan
Multitargeting Prodrugs that Release Oxaliplatin, Doxorubicin and Gemcitabine are Potent Inhibitors of Tumor Growth and Effective Inducers of Immunogenic Cell Death
2023 Sarkar, Amrita; Novohradsky, Vojtech; Maji, Moumita; Babu, Tomer; Markova, Lenka; Kostrhunova, Hana; Kasparkova, Jana; Gandin, Valentina; Brabec, Viktor; Gibson, Dan
1,2,4-Amino-triazine derivatives as pyruvate dehydrogenase kinase inhibitors: Synthesis and pharmacological evaluation
2023 Pecoraro, Camilla; DE FRANCO, Michele; Carbone, Daniela; Bassani, Davide; Pavan, Matteo; Cascioferro, Stella; Parrino, Barbara; Cirrincione, Girolamo; Dall'Acqua, Stefano; Moro, Stefano; Gandin, Valentina; Diana, Patrizia
Novel Silver Complexes Based on Phosphanes and Ester Derivatives of Bis(pyrazol-1-yl)acetate Ligands Targeting TrxR: New Promising Chemotherapeutic Tools Relevant to SCLC Management
2023 Pellei, Maura; Santini, Carlo; Bagnarelli, Luca; Caviglia, Miriam; Sgarbossa, Paolo; De Franco, Michele; Zancato, Mirella; Marzano, Cristina; Gandin, Valentina
Unusual tellurium(iv) mediated cyclisation diols into dihydroxazoles with potential anticancer activity
2023 D’Arcy, Kenneth; Schäfer, Tim; De Franco, Michele; Ricco, Raffaele; Gandin, Valentina; Sanz Miguel, Pablo J.; Montagner, Diego
Structural Manipulations of Marine Natural Products Inspire a New Library of 3-Amino-1,2,4-Triazine PDK Inhibitors Endowed with Antitumor Activity in Pancreatic Ductal Adenocarcinoma
2023 Carbone, Daniela; De Franco, Michele; Pecoraro, Camilla; Bassani, Davide; Pavan, Matteo; Cascioferro, Stella; Parrino, Barbara; Cirrincione, Girolamo; Dall’Acqua, Stefano; Sut, Stefania; Moro, Stefano; Gandin, Valentina; Diana, Patrizia
Pt(ii) and Pt(iv) complexes with a major component of royal jelly as innovative antitumor drug candidates
2023 Barbanente, Alessandra; Gandin, Valentina; Donati, Chiara; Pierro, Carmela Ilaria; Natile, Giovanni; Margiotta, Nicola
Synthesis and cytotoxicity studies of Cu(i) and Ag(i) complexes based on sterically hindered β-diketonates with different degrees of fluorination
2023 Pellei, Maura; Del Gobbo, Jo’; Caviglia, Miriam; Karade, Deepika V.; Gandin, Valentina; Marzano, Cristina; Noonikara Poyil, Anurag; Dias, H. V. Rasika; Santini, Carlo
Novel Biotinylated Cu(II)-Phenanthroline Complexes: 2D and 3D Cytotoxic Activity and Mechanistic Insight
2023 Barrett, Stephen; De Franco, Michele; Donati, Chiara; Marzano, Cristina; Gandin, Valentina; Montagner, Diego
Discovery of the 3-Amino-1,2,4-triazine-Based Library as Selective PDK1 Inhibitors with Therapeutic Potential in Highly Aggressive Pancreatic Ductal Adenocarcinoma
2023 Carbone, Daniela; DE FRANCO, Michele; Pecoraro, Camilla; Bassani, Davide; Pavan, Matteo; Cascioferro, Stella; Parrino, Barbara; Cirrincione, Girolamo; Dall’Acqua, Stefano; Moro, Stefano; Gandin, Valentina; Diana, Patrizia
Triiron Complex with N-Ferrocenyl Aminocarbyne Ligand Bridging a Diiron Core: DFT, Electrochemical, and Biological Insights
2023 Saviozzi, Chiara; Biancalana, Lorenzo; Funaioli, Tiziana; Bortoluzzi, Marco; De Franco, Michele; Guelfi, Massimo; Gandin, Valentina; Marchetti, Fabio
New tricyclic systems as photosensitizers towards triple negative breast cancer cells
2022 Barreca, Marilia; Ingarra, Angela Maria; Raimondi, Maria Valeria; Spanò, Virginia; Piccionello, Antonio Palumbo; De Franco, Michele; Menilli, Luca; Gandin, Valentina; Miolo, Giorgia; Barraja, Paola; Montalbano, Alessandra
Cu(I) and Cu(II) Complexes Based on Lonidamine-Conjugated Ligands Designed to Promote Synergistic Antitumor Effects
2022 Del Bello, Fabio; Pellei, Maura; Bagnarelli, Luca; Santini, Carlo; Giorgioni, Gianfabio; Piergentili, Alessandro; Quaglia, Wilma; Battocchio, Chiara; Iucci, Giovanna; Schiesaro, Irene; Meneghini, Carlo; Venditti, Iole; Ramanan, Nitya; De Franco, Michele; Sgarbossa, Paolo; Marzano, Cristina; Gandin, Valentina
Exploring the Antitumor Potential of Copper Complexes Based on Ester Derivatives of Bis(pyrazol-1-yl)acetate Ligands
2022 Pellei, Maura; Santini, Carlo; Bagnarelli, Luca; Battocchio, Chiara; Iucci, Giovanna; Venditti, Iole; Meneghini, Carlo; Amatori, Simone; Sgarbossa, Paolo; Marzano, Cristina; De Franco, Michele; Gandin, Valentina
Antiproliferative activity of nickel(II), palladium(II) and zinc(II) thiosemicarbazone complexes
2022 Carcelli, M.; Montalbano, S.; Rogolino, D.; Gandin, V.; Miglioli, F.; Pelosi, G.; Buschini, A.
Insight on pyrimido[5,4-g]indolizine and pyrimido[4,5-c]pyrrolo[1,2-a]azepine systems as promising photosensitizers on malignant cells
2022 Barreca, M; Ingarra, Am; Raimondi, Mv; Spanò, V; De Franco, M; Menilli, L; Gandin, V; Miolo, G; Barraja, P; Montalbano, A.
Preliminary Discovery of Small Molecule Inhibitors of Epidermal Growth Factor Receptor (EGFR) That Bind to the Extracellular Domain
2022 Di Liddo, Rosa; Verona, Marco; Vaccarin, Christian; Acquasaliente, Laura; Schrenk, Sandra; Piccione, Monica; Cenzi, Carola; De Franco, Michele; Dal Prà, Matteo; Ribaudo, Giovanni; Ferlin, Maria Grazia; Conconi, Maria Teresa; Chilin, Adriana; Gandin, Valentina; Marzaro, Giovanni
Decoding mechanism of action and sensitivity to drug candidates from integrated transcriptome and chromatin state
2022 Carraro, Caterina; Bonaguro, Lorenzo; Schulte-Schrepping, Jonas; Horne, Arik; Oestreich, Marie; Warnat-Herresthal, Stefanie; Helbing, Tim; De Franco, Michele; Haendler, Kristian; Mukherjee, Sach; Ulas, Thomas; Gandin, Valentina; Goettlich, Richard; Aschenbrenner, Anna C; Schultze, Joachim L; Gatto, Barbara
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