Sfoglia per Autore
4-[(4'-idrossifenil)sulfanil]-3-buten-2-one (HPSBO), un potenziale "lead" per losviluppo di agenti bifunzionali per la terapia mirata del melanoma
2007 Quintieri, Luigi; Rondina, Maria; Nassi, Alberto; Zorzin, M; Floreani, Maura; Rosato, Antonio; Rossi, CARLO RICCARDO; Ruzza, Paolo
Effect of 4-fluoro-l-proline on the sh3 binding affinitity
2007 Ruzza, Paolo; Rubini, Chiara; Siligardi, Gianfranco; Hussain, R; Calderan, Andrea; Guiotto, Adriano; Cesaro, Luca; Brunati, ANNA MARIA; Donella, Arianna
4-Fluoroproline derivative peptides: Effect on PPII conformation and SH3 affinity
2006 Ruzza, Paolo; Siligardi, G; Donella, Arianna; Calderan, Andrea; Hussain, R; Rubini, Chiara; Cesaro, Luca; Osler, A; Guiotto, Adriano; Pinna, Lorenzo; Borin, G.
Evaluation of tyrosine conformational restriction in PTK peptide substrates
2005 Ruzza, Paolo; Donella, Arianna; Calderan, Andrea; Osler, A; Rubini, Chiara; Menegazzo, Ileana; Biondi, Barbara; Cesaro, Luca; Guiotto, Adriano; Pinna, Lorenzo; Borin, Gianfranco
Effect of 4-S-fluoro-L-proline residue to enhance poly-proline type II helix binding conformation of SH3 binding peptides
2005 Ruzza, Paolo; Siligardi, Gianfranco; Donella, Arianna; Osler, A; Rubini, Chiara; Hussain, R; Brunati, ANNA MARIA; Calderan, Andrea; Guiotto, Adriano; Pinna, Lorenzo; Borin, Gianfranco
Binding interactions of phospho-Htc peptide to c-Fgr SH2 domain
2004 Ruzza, Paolo; A., Osler; DEL PIERO, Stefania; Donella, Arianna; Brunati, ANNA MARIA; Siligardi, Gianfranco; R., Hussain; Calderan, Andrea; Guiotto, Adriano; Pinna, Lorenzo; Borin, Gianfranco
Conformational constraints of Tyrosine in Protein Tyrosine Kinase substrates: Information about preferred bioactive side chain orientation
2003 Ruzza, Paolo; Calderan, Andrea; Donella, Arianna; Biondi, Barbara; Cesaro, Luca; A., Osler; S., Elardo; S., Guiotto; Pinna, Lorenzo; Borin, Gianfranco
Specific monitoring of Syk protein kinase activity by peptide substrates including constrained analogs of tyrosine
2002 Donella, Arianna; Ruzza, Paolo; Cesaro, Luca; Brunati, ANNA MARIA; Calderan, Andrea; Borin, Gianfranco; Pinna, Lorenzo
Antennapedia/HS1 chimeric phosphotyrosil peptide: conformational properties, binding capability to c-Fgr SH2 domain and cell permeability
2001 Ruzza, Paolo; Donella, Arianna; Calderan, Andrea; Brunati, ANNA MARIA; Massimino, MARIA LINA; Elardo, S.; Mattiazzo, A.; Pinna, Lorenzo; Borin, Gianfranco
Synthesis of selective substrates for Syk PTK
2001 Ruzza, Paolo; Calderan, Andrea; Donella, Arianna; Cesaro, Luca; Elardo, S; Pinna, Lorenzo; Borin, Gianfranco
Synthetic peptides as substrates or inhibitors of non-receptor protein tyrosine kinases
1999 Ruzza, Paolo; Donella, Arianna; Calderan, Andrea; Biondi, Barbara; Cesaro, Luca; Pinna, Lorenzo; Borin, Gianfranco
Nonhydrolyzable phosphotyrosine mimetic containing peptides interacting with Src SH2 domain
1999 Ruzza, Paolo; Donella, Arianna; Calderan, Andrea; Biondi, Barbara; Brunati, ANNA MARIA; Favretto, Donata; Pinna, Lorenzo; Borin, Gianfranco
Synthesis and biological activities of cyclic lactam peptides as substrates for non-receptor PTKs
1999 Ruzza, Paolo; Donella, Arianna; Calderan, Andrea; Biondi, Barbara; Pinna, Lorenzo; Borin, Gianfranco
Htc analogs of main autophosphorylation site of pp60src as selective substrates of Syk-PTK
1998 Ruzza, Paolo; Calderan, Andrea; Donella, Arianna; Pinna, Lorenzo; Borin, Gianfranco
Linear and cyclic peptides as substrates for lyn tyrosine kinase
1998 Ruzza, Paolo; Donella, Arianna; Calderan, Andrea; Zanotti, Giuseppe; Cesaro, Luca
An exploration of the effects of constraints on the phosphorylation of synthetic protein tyrosine kinase peptide substrates.
1996 Ruzza, Paolo; Donella, Arianna; Calderan, Andrea; Filippi, Bruno; Cesaro, Luca; Pinna, Lorenzo; Borin, Gianfranco
Linear and cyclic synthetic peptides related to the main autophosphorylation site of the Src tyrosine kinases as substrates and inhibitors of Lyn.
1995 Ruzza, Paolo; Calderan, Andrea; Filippi, Bruno; Biondi, Barbara; Donella, Arianna; Cesaro, Luca; Pinna, Lorenzo; Borin, Gianfranco
Synthetic Tyr-phosphopeptides as TPK inhibitors
1995 Ruzza, Paolo; Calderan, Andrea; Pavanetto, Martina; Donella, Arianna; Pinna, Lorenzo; Borin, Gianfranco
Synthetic Tyr-phospho and non-hydrolyzable phosphonopeptides as PTKs and TC-PTP inhibitors.
1995 Ruzza, Paolo; Donella, Arianna; Calderan, Andrea; Pavanetto, Martina; Cesaro, Luca; Pinna, Lorenzo; Borin, Gianfranco
Synthesis and conformational studies on peptides corresponding to a putative autophosphorylation site of abl TPK.
1993 Ruzza, Paolo; Calderan, Andrea; Filippi, Bruno; Donella, Arianna; Pinna, Lorenzo; Borin, Gianfranco
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