Sfoglia per Autore
A Broad anti-influenza hybrid small molecule that potently disrupts the interaction of polymerase acidic protein-basic protein 1 (PA-PB1) subunits
2015 Massari, Serena; Nannetti, Giulio; Desantis, Jenny; Muratore, Giulia; Sabatini, Stefano; Manfroni, Giuseppe; Mercorelli, Beatrice; Cecchetti, Violetta; Palu', Giorgio; Cruciani, Gabriele; Loregian, Arianna; Goracci, Laura; Tabarrini, Oriana
Optimization of Small-Molecule Inhibitors of Influenza Virus Polymerase: From Thiophene-3-Carboxamide to Polyamido Scaffolds
2014 Lepri, S; Nannetti, Giulio; Muratore, Giulia; Cruciani, G; Ruzziconi, R; Mercorelli, Beatrice; Palu', Giorgio; Loregian, Arianna; Goracci, L.
The 6-Aminoquinolone WC5 Inhibits Different Functions of the Immediate-Early 2 (IE2) Protein of Human Cytomegalovirus That Are Essential for Viral Replication.
2014 Mercorelli, Beatrice; Luganini, A; Muratore, G; Massari, S; Terlizzi, Me; Tabarrini, O; Gribaudo, G; Palu', Giorgio; Loregian, Arianna
Approaches for the generation of new anti-cytomegalovirus agents: identification of protein-protein interaction inhibitors and compounds against the HCMV IE2 protein.
2014 Mercorelli, Beatrice; Gribaudo, G; Palu', Giorgio; Loregian, Arianna
Antiviral strategies against influenza virus: towards new therapeutic approaches.
2014 Loregian, Arianna; Mercorelli, Beatrice; Nannetti, Giulio; Compagnin, Chiara; Palu', Giorgio
Structural investigation of cycloheptathiophene-3-carboxamide derivatives targeting influenza virus polymerase assembly.
2013 Massari, S; Nannetti, Giulio; Goracci, L; Sancineto, L; Muratore, Giulia; Sabatini, S; Manfroni, G; Mercorelli, Beatrice; Cecchetti, V; Facchini, M; Palu', Giorgio; Cruciani, G; Loregian, Arianna; Tabarrini, O.
Design, synthesis, and evaluation of WC5 analogues as inhibitors of human cytomegalovirus Immediate-Early 2 protein, a promising target for anti-HCMV treatment.
2013 Massari, S; Mercorelli, Beatrice; Sancineto, L; Sabatini, S; Cecchetti, V; Gribaudo, G; Palu', Giorgio; Pannecouque, C; Loregian, Arianna; Tabarrini, O.
Human Cytomegalovirus Inhibitor AL18 Also Possesses Activity against Influenza A and B Viruses.
2012 Muratore, Giulia; Mercorelli, Beatrice; Goracci, L; Cruciani, G; Digard, P; Palu', Giorgio; Loregian, Arianna
Small molecule inhibitors of influenza A and B viruses that act by disrupting subunit interactions of the viral polymerase.
2012 Muratore, Giulia; Goracci, L; Mercorelli, Beatrice; Foeglein, Á; Digard, P; Cruciani, G; Palu', Giorgio; Loregian, Arianna
The Human Cytomegalovirus DNA Polymerase Processivity Factor UL44 is Modified by SUMO in a DNA-dependent manner
2012 Sinigalia, Elisa; Alvisi, Gualtiero; Segré, Cv; Mercorelli, Beatrice; Muratore, Giulia; Winkler, M; Hsiao H., H; Urlaub, H; Ripalti, A; Chiocca, S; Palu', Giorgio; Loregian, Arianna
Early inhibitors of human cytomegalovirus: State-of-art and therapeutic perspectives.
2011 Mercorelli, Beatrice; Lembo, D; Palu', Giorgio; Loregian, Arianna
Sulfated Derivatives of Escherichia coli K5 Polysaccharide are Potent Inhibitors of Human Cytomegalovirus.
2010 Mercorelli, Beatrice; Oreste, P; Sinigalia, Elisa; Muratore, Giulia; Lembo, D; Palu', Giorgio; Loregian, Arianna
The 6-Aminoquinolone WC5 Inhibits Human Cytomegalovirus Replication at an Early Stage by Interfering with the Transactivating Activity of Viral Immediate-Early 2 Protein
2010 Loregian, Arianna; Mercorelli, Beatrice; Muratore, Giulia; Sinigalia, Elisa; Pagni, Silvana; Massari, S; Gribaudo, G; Gatto, Barbara; Palumbo, Manlio; Tabarrini, O; Cecchetti, V; Palu', Giorgio
Composition and methods for the treatment of pathological condition associated with cytomegalovirus infection.
2010 Loregian, Arianna; Palu', Giorgio; Mercorelli, Beatrice; Tabarrini, O.; Cecchetti, V.
Caratterizzazione di nuovi composti antivirali contro il citomegalovirus umano e studio del meccanismo di neuropatogenocità nel herpesvirus equino di tipo 1
2009 Mercorelli, Beatrice
A 6-Aminoquinolone Compound, WC5, with Potent and Selective Anti-Human Cytomegalovirus Activity
2009 Mercorelli, Beatrice; Muratore, Giulia; Sinigalia, Elisa; Tabarrini, O; Biasolo, MARIA-ANGELA; Cecchetti, V; Palu', Giorgio; Loregian, Arianna
Role of homodimerization of human cytomegalovirus DNA polymerase accessory protein UL44 in origin-dependent DNA replication in cells.
2008 Sinigalia, Elisa; Alvisi, Gualtiero; Mercorelli, Beatrice; Coen, Dm; Pari, Gs; Jans, Da; Ripalti, A; Palu', Giorgio; Loregian, Arianna
Human cytomegalovirus DNA replication: antiviral targets and drugs.
2008 Mercorelli, Beatrice; Sinigalia, Elisa; Loregian, Arianna; Palu', Giorgio
A point mutation in a herpesvirus polymerase determines neuropathogenicity.
2007 Goodman, L. B.; Loregian, Arianna; Perkins, G. A.; Nugent, J; Buckles, E. L.; Mercorelli, Beatrice; Kydd, J. H.; Palu', Giorgio; Smith, K. C.; Osterrieder, N; DAVIS POYNTER, N.
Binding parameters and thermodynamics of the interaction of the human cytomegalovirus DNA polymerase accessory protein, UL44, with DNA: implications for the processivity mechanism
2007 Loregian, Arianna; Sinigalia, Elisa; Mercorelli, Beatrice; Palu', Giorgio; Coen, Dm
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