Sfoglia per Autore
Design, Synthesis, and Biological Evaluation of 6-Substituted Thieno[3,2- d]pyrimidine Analogues as Dual Epidermal Growth Factor Receptor Kinase and Microtubule Inhibitors
2019 Romagnoli, R.; Prencipe, F.; Oliva, P.; Baraldi, S.; Baraldi, P. G.; Schiaffino Ortega, S.; Chayah, M.; Kimatrai Salvador, M.; Lopez-Cara, L. C.; Brancale, A.; Ferla, S.; Hamel, E.; Ronca, R.; Bortolozzi, R.; Mariotto, E.; Mattiuzzo, E.; Viola, G.
Potent In Vitro and In Vivo Anticancer Activity of New Bipyridine and Bipyrimidine Gold (III) Dithiocarbamate Derivatives
2019 Altaf, Muhammad; Casagrande, Naike; Mariotto, Elena; Baig, Nadeem; Kawde, Abdel-Nasser; Corona, Giuseppe; Larcher, Roberto; Borghese, Cinzia; Pavan, Claudia; Seliman, Adam; Aldinucci, Donatella; Isab, Anvarhusein
SYK targeting represents a potential therapeutic option for relapsed resistant pediatric ETV6-RUNX1 B-acute lymphoblastic leukemia patients
2019 Serafin, V.; Porcu, E.; Cortese, G.; Mariotto, E.; Veltri, G.; Bresolin, S.; Basso, G.; Accordi, B.
Lead optimization-hit expansion of new asymmetrical pyridinium/quinolinium compounds as choline kinase α1 inhibitors
2018 Rubbini, Gianluca; Buades-Martín, Ana Begoña; Kimatrai-Salvador, María; Entrena, Antonio; Gallo-Mezo, Miguel Ángel; Ríos-Marco, Pablo; Marco, Carmen; Mattiuzzo, Elena; Bortolozzi, Roberta; Mariotto, Elena; Greco, Francesco Antonio; Macchiarulo, Antonio; Carrasco-Jiménez, María Paz; Viola, Giampietro; López-Cara, Luisa Carlota
Choline kinase alpha inhibition by EB-3D triggers cellular senescence, reduces tumor growth and metastatic dissemination in breast cancer
2018 Mariotto, Elena; Viola, Giampietro; Ronca, Roberto; Persano, Luca; Aveic, Sanja; Bhujwalla, Zaver M.; Mori, Noriko; Accordi, Benedetta; Serafin, Valentina; López-Cara, Luisa Carlota; Bortolozzi, Roberta
AKR1C enzymes sustain therapy resistance in paediatric T-ALL
2018 Bortolozzi, Roberta; Bresolin, Silvia; Rampazzo, Elena; Paganin, Maddalena; Maule, Francesca; Mariotto, Elena; Boso, Daniele; Minuzzo, Sonia; Agnusdei, Valentina; Viola, Giampietro; Te Kronnie, Geertruy; Cazzaniga, Giovanni; Basso, Giuseppe; Persano, Luca
EB-3D a novel choline kinase inhibitor induces deregulation of the AMPK-mTOR pathway and apoptosis in leukemia T-cells
2018 Mariotto, Elena; Bortolozzi, Roberta; Volpin, Ilaria; Carta, Davide; Serafin, Valentina; Accordi, Benedetta; Basso, Giuseppe; Navarro, Pilar Luque; López-Cara, Luisa Carlota; Viola, Giampietro
TP-0903 inhibits neuroblastoma cell growth and enhances the sensitivity to conventional chemotherapy
2018 Aveic, Sanja; Corallo, Diana; Porcã¹, Elena; Pantile, Marcella; Boso, Daniele; Zanon, Carlo; Viola, Giampietro; Sidarovich, Viktoryia; Mariotto, Elena; Quattrone, Alessandro; Basso, Giuseppe; Tonini, Gian Paolo
In vitro and in vivo antitumor activity of new choline kinase inhibitor: a pharmacological strategy for breast cancer and leukemia treatment.
2017 Mariotto, Elena
Synthesis and Biological Evaluation of 2-Methyl-4,5-Disubstituted Oxazoles as a Novel Class of Highly Potent Antitubulin Agents
2017 Romagnoli, Romeo; Baraldi, Pier Giovanni; Prencipe, Filippo; Oliva, Paola; Baraldi, Stefania; Salvador, Maria Kimatrai; Lopez-Cara, Luisa Carlota; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Ronca, Roberto; Bortolozzi, Roberta; Mariotto, Elena; Porcã¹, Elena; Basso, Giuseppe; Viola, Giampietro
Design and synthesis of potent in vitro and in vivo anticancer agents based on 1-(3',4',5'-trimethoxyphenyl)-2-Aryl-1H-imidazole
2016 Romagnoli, Romeo; Baraldi, Pier Giovanni; Prencipe, Filippo; Oliva, Paola; Baraldi, Stefania; Tabrizi, Mojgan Aghazadeh; Lopez-Cara, Luisa Carlota; Ferla, Salvatore; Brancale, Andrea; Hamel, Ernest; Ronca, Roberto; Bortolozzi, Roberta; Mariotto, Elena; Basso, Giuseppe; Viola, Giampietro
Design, synthesis, crystallization and biological evaluation of new symmetrical biscationic compounds as selective inhibitors of human Choline Kinase α1 (ChoKα1)
2016 Schiaffino-Ortega, Santiago; Baglioni, Eleonora; Mariotto, Elena; Bortolozzi, Roberta; Serrán-Aguilera, Luciá; Riós-Marco, Pablo; Carrasco-Jimenez, M. Paz; Gallo, Miguel A.; Hurtado-Guerrero, Ramon; Marco, Carmen; Basso, Giuseppe; Viola, Giampietro; Entrena, Antonio; López-Cara, Luisa Carlota
HLA Class II Antibody Activation of Endothelial Cells Promotes Th17 and Disrupts Regulatory T Lymphocyte Expansion
2016 Lion, J.; Taflin, C.; Cross, A. R.; Robledo-Sarmiento, M.; Mariotto, E.; Savenay, A.; Carmagnat, M.; Suberbielle, C.; Charron, D.; Haziot, A.; Glotz, D.; Mooney, N.
New more polar symmetrical bipyridinic compounds: new strategy for the inhibition of choline kinase α1
2015 Castro-Navas, Francisco Fermín; Schiaffino-Ortega, Santiago; Carrasco-Jimenez, María Paz; Ríos-Marco, Pablo; Marco, Carmen; Espinosa, Antonio; Gallo, Miguel Angel; Mariotto, Elena; Basso, Giuseppe; Viola, Giampietro; Entrena-Guadix, Antonio; López-Cara, Luisa Carlota
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile