BORTOLOZZI, ROBERTA
BORTOLOZZI, ROBERTA
Dipartimento di Salute della Donna e del Bambino - SDB
Synthesis and in vitro evaluation of 3H-pyrrolo[3,2-f[quinolin-9-one derivatives that show potent and selective anti-leukemic activity
2010 Ferlin, MARIA GRAZIA; Bortolozzi, Roberta; Brun, Paola; Castagliuolo, Ignazio; Hamel, E; Basso, Giuseppe; Viola, Giampietro
Synthesis and Evaluation of 1,5-Disubstituted Tetrazoles as Rigid Analogues of Combretastatin A-4 with Potent Antiproliferative and Antitumor Activity
2012 Romeo, Romagnoli; Pier Giovanni Baraldi, ; Maria Kimatrai Salvador, ; Delia, Preti; Mojgan Aghazadeh Tabrizi, ; Andrea, Brancale; Xian Hua Fu, ; Jun, Li; Su Zhan Zhang, ; Ernest, Hamel; Bortolozzi, Roberta; Basso, Giuseppe; Viola, Giampietro
MG-2477, a new tubulin inhibitor, induces autophagy through inhibition of the Akt/mTOR pathway and delayed apoptosis in A549 cells.
2012 Viola, Giampietro; Bortolozzi, Roberta; Hamel, E; Moro, Stefano; Brun, Paola; Castagliuolo, Ignazio; Ferlin, MARIA GRAZIA; Basso, Giuseppe
Synthesis and biological evaluation of 2-substituted-4-(3',4',5'-trimethoxyphenyl)-5-aryl thiazoles as anticancer agents.
2012 Romagnoli, R; Baraldi, Pg; Salvador, Mk; Camacho, Me; Preti, D; Tabrizi, Ma; Bassetto, M; Brancale, A; Hamel, E; Bortolozzi, Roberta; Basso, Giuseppe; Viola, G.
Discovery of a novel class of anti-proliferative pyrrolo[3,2-f]quinolin-9-ones characterized by interfering with both PI3K-Akt-mTOR signalling and microtubule assembling
2012 Ferlin, MARIA GRAZIA; Viola, Giampietro; Bortolozzi, Roberta; Carta, Davide; Hamel, E.; Moro, Stefano; Basso, Giuseppe
Synthesis and biological evaluation of 2-substituted-4-(3â²,4â², 5â²-trimethoxyphenyl)-5-aryl thiazoles as anticancer agents
2012 Romagnoli, Romeo; Baraldi, Pier Giovanni; Salvador, Maria Kimatrai; Camacho, M. Encarnacion; Preti, Delia; Tabrizi, Mojgan Aghazadeh; Bassetto, Marcella; Brancale, Andrea; Hamel, Ernest; Bortolozzi, Roberta; Basso, Giuseppe; Viola, Giampietro
Study of the mechanism of action of new molecules endowed with antitumoral activity
2012 Bortolozzi, Roberta
TR-644 a novel potent tubulin binding agent induces impairment of endothelial cells function and inhibits angiogenesis
2013 Elena, Porcù; Viola, Giampietro; Bortolozzi, Roberta; Persano, Luca; Stefania, Mitola; Roberto, Ronca; Marco, Presta; Romeo, Romagnoli; Pier Giovanni, Baraldi; Basso, Giuseppe
Synthesis and Biological Evaluation of 2-(Alkoxycarbonyl)-3-Anilinobenzo[b]thiophenes and Thieno[2,3-b]pyridines as New Potent Anticancer Agents.
2013 Romagnoli, R; Baraldi, Pg; Kimatrai Salvador, M; Preti, D; Aghazadeh Tabrizi, M; Bassetto, M; Brancale, A; Hamel, E; Castagliuolo, Ignazio; Bortolozzi, Roberta; Basso, Giuseppe; Viola, Giampietro
Azolylmethyl-pyrroloquinolines as non steroidal aromatase inhibitors
2013 Ferlin, MARIA GRAZIA; Carta, Davide; Bortolozzi, Roberta; Ghodsi, R.; Chimento, A.; Pezzi, V.; Moro, Stefano; Basso, Giuseppe; Viola, Giampietro
Design, synthesis and SARs of azolylmethyl-pyrroloquinolines as non steroidal aromatase inhibitors, NPCF7
2013 Carta, Davide; Ferlin, MARIA GRAZIA; Bortolozzi, Roberta; Ghodsi, R.; Chimento, A.; Pezzi, V.; Moro, Stefano; Basso, Giuseppe; Viola, Giampietro
Design, synthesis and biological evaluation of 3,5-disubstituted 2-amino thiophene derivatives as a novel class of antitumor agents.
2013 Romagnoli, R; Baraldi, Pg; Lopez Cara, C; Salvador, Mk; Preti, D; Tabrizi, Ma; Balzarini, J; Nussbaumer, P; Bassetto, M; Brancale, A; Fu, Xh; Yang, Gao; Li, J; Zhang, Sz; Hamel, E; Bortolozzi, Roberta; Basso, Giuseppe; Viola, G.
Design and synthesis of azolylmethyl-pyrroloquinolines as potent and selective non steroidal CYP19 inhibitors
2013 Carta, Davide; Bortolozzi, Roberta; Ghodsi, R.; Chimento, A.; Pezzi, V.; Moro, Stefano; Hanke, N.; Hartmann, R.; Basso, Giuseppe; Viola, Giampietro; Ferlin, MARIA GRAZIA
Design, Synthesis, and Structure–Activity Relationships of Azolylmethylpyrroloquinolines as Nonsteroidal Aromatase Inhibitors
2013 Ferlin, MARIA GRAZIA; Carta, Davide; Bortolozzi, Roberta; Razieh, Ghodsi; Adele, Chimento; Vincenzo, Pezzi; Moro, Stefano; Nina, Hanke; Rolf W., Hartmann; Basso, Giuseppe; Viola, Giampietro
9-(4-Dimethylaminophenyl)benzo[b]quinolizinium: A Near-Infrared Fluorophore for the Multicolor Analysis of Proteins and Nucleic Acids in Living Cells
2013 Bortolozzi, Roberta; Heiko, Ihmels; Laura, Thomas; Maoqun, Tian; Viola, Giampietro
Concise Synthesis and Biological Evaluation of 2-Aroyl-5-Amino Benzo[ b ]thiophene Derivatives As a Novel Class of Potent Antimitotic Agents
2013 Romagnoli, Romeo; Baraldi, Pier Giovanni; Lopez-Cara, Carlota; Preti, Delia; Aghazadeh Tabrizi, Mojgan; Balzarini, Jan; Bassetto, Marcella; Brancale, Andrea; Fu, Xian-Hua; Gao, Yang; Li, Jun; Zhang, Su-Zhan; Hamel, Ernest; Bortolozzi, Roberta; Basso, Giuseppe; Viola, Giampietro
Natural daucane esters induces apoptosis in leukaemic cells through ROS production
2014 Dall'Acqua, Stefano; Linardi, M. A.; Bortolozzi, Roberta; Clauser, Maria; Marzocchini, S.; Maggi, F.; Nicoletti, M.; Innocenti, Gabbriella; Basso, Giuseppe; Viola, Giampietro
Synthesis, biological evaluation and molecular docking studies of trans-indole-3-acrylamide derivatives, a new class of tubulin polymerization inhibitors
2014 Sultan Nacak, Baytas; Nazan, Inceler; Akın, Yılmaz; Abdurrahman, Olgac; Sevda, Menevse; Erden, Banoglu; Ernest, Hamel; Bortolozzi, Roberta; Viola, Giampietro
Hemiasterlin analogues incorporating an aromatic, and heterocyclic type C-terminus: Design, synthesis and biological evaluation
2014 Lesma, Giordano; Sacchetti, Alessandro; Bai, Rouli; Basso, Giuseppe; Bortolozzi, Roberta; Hamel, Ernest; Silvani, Alessandra; Vaiana, Nadia; Viola, Giampietro
Discovery of MG-2603 with in vitro potent antiproliferative activity by interfering with kinases and tubulin polymerisation
2014 Carta, Davide; Ferlin, MARIA GRAZIA; Bortolozzi, Roberta; Moro, Stefano; Viola, Giampietro