MORIZZO, ERIKA
MORIZZO, ERIKA
2-Phenylpyrazolo[4,3-d]pyrimidin-7-one as a New Scaffold To Obtain Potent and Selective Human A(3) Adenosine Receptor Antagonists: New Insights into the Receptor-Antagonist Recognition
2009 Lenzi, O; Colotta, V; Catarzi, D; Varano, F; Poli, D; Filacchioni, G; Varani, K; Vincenzi, F; Borea, Pa; Paoletta, Silvia; Morizzo, Erika; Moro, Stefano
4-amido-2-aryl-1,2,4-triazolo[4,3-a]quinoxalin-1-ones as new potent and selective human A(3) adenosine receptor antagonists. synthesis, pharmacological evaluation, and ligand-receptor modeling studies
2006 Lenzi, O; Colotta, V; Catarzi, D; Varano, F; Filacchioni, G; Martini, C; Trincavelli, L; Ciampi, O; Varani, K; Marighetti, F; Morizzo, Erika; Moro, Stefano
A novel class of pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidines as A(3) adenosine receptor antagonists
2010 Federico, S; Spalluto, G; Klotz, Kn; Cacciari, B; Moro, Stefano; Morizzo, Erika
G Protein-Coupled Receptors as Potential Drug Target: From Receptor Topology to Rational Drug Design, an in-silico Approach
2009 Morizzo, Erika
Human A(3) Adenosine Receptor as Versatile G Protein-Coupled Receptor Example to Validate the Receptor Homology Modeling Technology
2009 Morizzo, Erika; Federico, S; Spalluto, G; Moro, Stefano
New 2-arylpyrazolo[3,4-c]quinoline derivatives as potent and selective human A(3) adenosine receptor antagonists. Synthesis, pharmacological evaluation, and ligand-receptor modeling studies
2007 Colotta, V; Catarzi, D; Varano, F; Capelli, F; Lenzi, O; Filacchioni, G; Martini, C; Trincavelli, L; Ciampi, O; Pugliese, Am; Pedata, F; Schiesaro, A; Morizzo, Erika; Moro, Stefano
Pyrazolo-triazolo-pyrimidines as adenosine receptor antagonists: Effect of the N-5 bond type on the affinity and selectivity at the four adenosine receptor subtypes
2008 Bolcato, C; Cusan, C; Pastorin, G; Spalluto, G; Cacciari, B; Klotz, Kn; Morizzo, Erika; Moro, Stefano
Pyrido[2,3-e]-1,2,4-triazolo[4,3-a]pyrazin-1-one as a New Scaffold To Develop Potent and Selective Human A(3) Adenosine Receptor Antagonists. Synthesis, Pharmacological Evaluation, and Ligand-Receptor Modeling Studies
2009 Colotta, V; Lenzi, O; Catarzi, D; Varano, F; Filacchioni, G; Martini, C; Trincavelli, L; Ciampi, O; Pugliese, Am; Traini, C; Pedata, F; Morizzo, Erika; Moro, Stefano
Scouting human A(3) adenosine receptor antagonist binding mode using a molecular simplification approach: From triazoloquinoxaline to a pyrimidine skeleton as a key study
2007 Morizzo, Erika; Capelli, F; Lenzi, O; Catarzi, D; Varano, F; Filacchioni, G; Vincenzi, F; Varani, K; Borea, Pa; Colotta, V; Moro, Stefano
Synthesis, ligand-receptor modeling studies and pharmacological evaluation of novel 4-modified-2-aryl-1,2,4-triazolo[4,3-a]quinoxalin-1-one derivatives as potent and selective human A(3) adenosine receptor antagonists
2008 Colotta, V; Catarzi, D; Varano, F; Lenzi, O; Filacchioni, G; Martini, C; Trincavelli, L; Ciampi, O; Traini, C; Pugliese, Am; Pedata, F; Morizzo, Erika; Moro, Stefano