Sfoglia per Autore
Design and synthesis of potent in vitro and in vivo anticancer agents based on 1-(3',4',5'-trimethoxyphenyl)-2-Aryl-1H-imidazole
2016 Romagnoli, Romeo; Baraldi, Pier Giovanni; Prencipe, Filippo; Oliva, Paola; Baraldi, Stefania; Tabrizi, Mojgan Aghazadeh; Lopez-Cara, Luisa Carlota; Ferla, Salvatore; Brancale, Andrea; Hamel, Ernest; Ronca, Roberto; Bortolozzi, Roberta; Mariotto, Elena; Basso, Giuseppe; Viola, Giampietro
Design, synthesis, crystallization and biological evaluation of new symmetrical biscationic compounds as selective inhibitors of human Choline Kinase α1 (ChoKα1)
2016 Schiaffino-Ortega, Santiago; Baglioni, Eleonora; Mariotto, Elena; Bortolozzi, Roberta; Serrán-Aguilera, Luciá; Riós-Marco, Pablo; Carrasco-Jimenez, M. Paz; Gallo, Miguel A.; Hurtado-Guerrero, Ramon; Marco, Carmen; Basso, Giuseppe; Viola, Giampietro; Entrena, Antonio; López-Cara, Luisa Carlota
Vascular disrupting activity of combretastatin analogues
2016 Porcù, Elena; Salvador, Alessia; Primac, Irina; Mitola, Stefania; Ronca, Roberto; Ravelli, Cosetta; Bortolozzi, Roberta; Vedaldi, Daniela; Romagnoli, Romeo; Basso, Giuseppe; Viola, Giampietro
Complementary isonitrile-based multicomponent reactions for the synthesis of diversified cytotoxic hemiasterlin analogues
2015 Lesma, Giordano; Bassanini, Ivan; Bortolozzi, Roberta; Colletto, Chiara; Bai, Ruoli; Hamel, Ernest; Meneghetti, Fiorella; Rainoldi, Giulia; Stucchi, Mattia; Sacchetti, Alessandro; Silvani, Alessandra; Viola, Giampietro
FOXO3a and posttranslational modifications mediate glucocorticoid sensitivity in B-ALL
2015 Consolaro, Francesca; Ghaem-Maghami, Sadaf; Bortolozzi, Roberta; Zona, Stefania; Khongkow, Mattaka; Basso, Giuseppe; Viola, Giampietro; Lam, Eric W. -F.
Novel 3-Substituted 7-Phenylpyrrolo[3,2-f]quinolin-9(6H)-ones as Single Entities with Multitarget Antiproliferative Activity
2015 Carta, Davide; Bortolozzi, Roberta; Hamel, Ernest; Basso, Giuseppe; Moro, Stefano; Viola, Giampietro; Ferlin, MARIA GRAZIA
Discovery of MG-2603 with in vitro potent antiproliferative activity by interfering with kinases and tubulin polymerisation
2015 Carta, Davide; Ferlin, MARIA GRAZIA; Bortolozzi, Roberta; Moro, Stefano; Viola, Giampietro
Design, synthesis, in vitro, and in vivo anticancer and antiangiogenic activity of novel 3-arylaminobenzofuran derivatives targeting the colchicine site on tubulin
2015 Romeo, Romagnoli; Pier Giovanni Baraldi, ; Maria Kimatrai Salvador, ; Filippo, Prencipe; Carlota Lopez Cara, ; Santiago Schiaffino Ortega, ; Andrea, Brancale; Ernest, Hamel; Castagliuolo, Ignazio; Stefania, Mitola; Roberto, Ronca; Bortolozzi, Roberta; Elena, Porcù; Basso, Giuseppe; Viola, Giampietro
Design, synthesis and biological evaluation of 3,5-disubstituted 2-amino thiophene derivatives as a novel class of antitumor agents
2015 Romagnoli, Romeo; Baraldi, Pier Giovanni; Lopez-Cara, Carlota; Salvador, Maria Kimatrai; Preti, Delia; Tabrizi, Mojgan Aghazadeh; Balzarini, Jan; Nussbaumer, Peter; Bassetto, Marcella; Brancale, Andrea; Fu, Xian-Hua; Yang-Gao, Null; Li, Jun; Zhang, Su-Zhan; Hamel, Ernest; Bortolozzi, Roberta; Basso, Giuseppe; Viola, Giampietro
Hemiasterlin analogues incorporating an aromatic, and heterocyclic type C-terminus: design, synthesis and biological evaluation
2014 Lesma, Giordano; Sacchetti, Alessandro; Bai, Rouli; Basso, Giuseppe; Bortolozzi, Roberta; Hamel, Ernest; Silvani, Alessandra; Vaiana, Nadia; Viola, Giampietro
Selective ratiometric detection of H2O2in water and in living cells with boronobenzo[b]quinolizinium derivatives
2014 Bortolozzi, Roberta; Sebastian von, Gradowski; Heiko, Ihmels; Katy, Schäfer; Viola, Giampietro
Discovery of MG-2603 with in vitro potent antiproliferative activity by interfering with kinases and tubulin polymerisation
2014 Carta, Davide; Ferlin, MARIA GRAZIA; Bortolozzi, Roberta; Moro, Stefano; Viola, Giampietro
Natural daucane esters induces apoptosis in leukaemic cells through ROS production
2014 Dall'Acqua, Stefano; Linardi, M. A.; Bortolozzi, Roberta; Clauser, Maria; Marzocchini, S.; Maggi, F.; Nicoletti, M.; Innocenti, Gabbriella; Basso, Giuseppe; Viola, Giampietro
Synthesis, biological evaluation and molecular docking studies of trans-indole-3-acrylamide derivatives, a new class of tubulin polymerization inhibitors
2014 Sultan Nacak, Baytas; Nazan, Inceler; Akın, Yılmaz; Abdurrahman, Olgac; Sevda, Menevse; Erden, Banoglu; Ernest, Hamel; Bortolozzi, Roberta; Viola, Giampietro
A novel copper(I) complex induces ER-stress-mediated apoptosis and sensitizes B-acute lymphoblastic leukemia cells to chemotherapeutic agents
2014 Bortolozzi, Roberta; Viola, G.; Porcù, E.; Consolaro, Francesca; Marzano, Cristina; Pellei, M.; Gandin, Valentina; Basso, Giuseppe
TR-644 a novel potent tubulin binding agent induces impairment of endothelial cells function and inhibits angiogenesis
2013 Elena, Porcù; Viola, Giampietro; Bortolozzi, Roberta; Persano, Luca; Stefania, Mitola; Roberto, Ronca; Marco, Presta; Romeo, Romagnoli; Pier Giovanni, Baraldi; Basso, Giuseppe
Synthesis and Biological Evaluation of 2-(Alkoxycarbonyl)-3-Anilinobenzo[b]thiophenes and Thieno[2,3-b]pyridines as New Potent Anticancer Agents.
2013 Romagnoli, R; Baraldi, Pg; Kimatrai Salvador, M; Preti, D; Aghazadeh Tabrizi, M; Bassetto, M; Brancale, A; Hamel, E; Castagliuolo, Ignazio; Bortolozzi, Roberta; Basso, Giuseppe; Viola, Giampietro
Design, synthesis and biological evaluation of 3,5-disubstituted 2-amino thiophene derivatives as a novel class of antitumor agents.
2013 Romagnoli, R; Baraldi, Pg; Lopez Cara, C; Salvador, Mk; Preti, D; Tabrizi, Ma; Balzarini, J; Nussbaumer, P; Bassetto, M; Brancale, A; Fu, Xh; Yang, Gao; Li, J; Zhang, Sz; Hamel, E; Bortolozzi, Roberta; Basso, Giuseppe; Viola, G.
Design, Synthesis, and Structure–Activity Relationships of Azolylmethylpyrroloquinolines as Nonsteroidal Aromatase Inhibitors
2013 Ferlin, MARIA GRAZIA; Carta, Davide; Bortolozzi, Roberta; Razieh, Ghodsi; Adele, Chimento; Vincenzo, Pezzi; Moro, Stefano; Nina, Hanke; Rolf W., Hartmann; Basso, Giuseppe; Viola, Giampietro
Azolylmethyl-pyrroloquinolines as non steroidal aromatase inhibitors
2013 Ferlin, MARIA GRAZIA; Carta, Davide; Bortolozzi, Roberta; Ghodsi, R.; Chimento, A.; Pezzi, V.; Moro, Stefano; Basso, Giuseppe; Viola, Giampietro
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