Sfoglia per Autore
Design, synthesis and biological evaluation of novel vicinal diaryl-substituted 1H-Pyrazole analogues of combretastatin A-4 as highly potent tubulin polymerization inhibitors
2019 Romagnoli, R.; Oliva, P.; Salvador, M. K.; Camacho, M. E.; Padroni, C.; Brancale, A.; Ferla, S.; Hamel, E.; Ronca, R.; Grillo, E.; Bortolozzi, R.; Rruga, F.; Mariotto, E.; Viola, G.
Identification of novel indole derivatives acting as inhibitors of the Keap1-Nrf2 interaction
2019 Cosimelli, Barbara; Greco, Giovanni; Laneri, Sonia; Novellino, Ettore; Sacchi, Antonia; Amendola, Giorgio; Cosconati, Sandro; Bortolozzi, Roberta; Viola, Giampietro
Evaluating the effects of fluorine on biological properties and metabolic stability of some antitubulin 3-substituted 7-phenyl-pyrroloquinolinones
2019 Bortolozzi, R.; Carta, D.; Dal Pra, M.; Antoniazzi, G.; Mattiuzzo, E.; Sturlese, M.; Di Paolo, V.; Calderan, L.; Moro, S.; Hamel, E.; Quintieri, L.; Ronca, R.; Viola, G.; Ferlin, M. G.
Synthesis, in vitro and in vivo biological evaluation of substituted 3-(5-imidazo[2,1-b]thiazolylmethylene)-2-indolinones as new potent anticancer agents
2019 Morigi, R.; Locatelli, A.; Leoni, A.; Rambaldi, M.; Bortolozzi, R.; Mattiuzzo, E.; Ronca, R.; Maccarinelli, F.; Hamel, E.; Bai, R.; Brancale, A.; Viola, G.
Design, Synthesis, and Biological Evaluation of 6-Substituted Thieno[3,2- d]pyrimidine Analogues as Dual Epidermal Growth Factor Receptor Kinase and Microtubule Inhibitors
2019 Romagnoli, R.; Prencipe, F.; Oliva, P.; Baraldi, S.; Baraldi, P. G.; Schiaffino Ortega, S.; Chayah, M.; Kimatrai Salvador, M.; Lopez-Cara, L. C.; Brancale, A.; Ferla, S.; Hamel, E.; Ronca, R.; Bortolozzi, R.; Mariotto, E.; Mattiuzzo, E.; Viola, G.
Choline kinase alpha inhibition by EB-3D triggers cellular senescence, reduces tumor growth and metastatic dissemination in breast cancer
2018 Mariotto, Elena; Viola, Giampietro; Ronca, Roberto; Persano, Luca; Aveic, Sanja; Bhujwalla, Zaver M.; Mori, Noriko; Accordi, Benedetta; Serafin, Valentina; López-Cara, Luisa Carlota; Bortolozzi, Roberta
AKR1C enzymes sustain therapy resistance in paediatric T-ALL
2018 Bortolozzi, Roberta; Bresolin, Silvia; Rampazzo, Elena; Paganin, Maddalena; Maule, Francesca; Mariotto, Elena; Boso, Daniele; Minuzzo, Sonia; Agnusdei, Valentina; Viola, Giampietro; Te Kronnie, Geertruy; Cazzaniga, Giovanni; Basso, Giuseppe; Persano, Luca
Targeting tubulin polymerization by novel 7-aryl-pyrroloquinolinones: Synthesis, biological activity and SARs
2018 Bortolozzi, Roberta; Mattiuzzo, Elena; Dal Pra, Matteo; Sturlese, Mattia; Moro, Stefano; Hamel, Ernest; Carta, Davide; Viola, Giampietro; Ferlin, Maria Grazia
Phytosterol and γ-Oryzanol Conjugates: Synthesis and Evaluation of their Antioxidant, Antiproliferative, and Anticholesterol Activities
2018 Lesma, Giordano; Luraghi, Andrea; Bavaro, Teodora; Bortolozzi, Roberta; Rainoldi, Giulia; Roda, Gabriella; Viola, Giampietro; Ubiali, Daniela; Silvani, Alessandra
EB-3D a novel choline kinase inhibitor induces deregulation of the AMPK-mTOR pathway and apoptosis in leukemia T-cells
2018 Mariotto, Elena; Bortolozzi, Roberta; Volpin, Ilaria; Carta, Davide; Serafin, Valentina; Accordi, Benedetta; Basso, Giuseppe; Navarro, Pilar Luque; López-Cara, Luisa Carlota; Viola, Giampietro
Ribociclib, a Cdk4/Cdk6 kinase inhibitor, enhances glucocorticoid sensitivity in B-acute lymphoblastic leukemia (B-All)
2018 Bortolozzi, Roberta; Mattiuzzo, Elena; Trentin, Luca; Accordi, Benedetta; Basso, Giuseppe; Viola, Giampietro
Lead optimization-hit expansion of new asymmetrical pyridinium/quinolinium compounds as choline kinase α1 inhibitors
2018 Rubbini, Gianluca; Buades-Martín, Ana Begoña; Kimatrai-Salvador, María; Entrena, Antonio; Gallo-Mezo, Miguel Ángel; Ríos-Marco, Pablo; Marco, Carmen; Mattiuzzo, Elena; Bortolozzi, Roberta; Mariotto, Elena; Greco, Francesco Antonio; Macchiarulo, Antonio; Carrasco-Jiménez, María Paz; Viola, Giampietro; López-Cara, Luisa Carlota
3-Aryl/Heteroaryl-5-amino-1-(3',4',5'-trimethoxybenzoyl)-1,2,4-triazoles as antimicrotubule agents. Design, synthesis, antiproliferative activity and inhibition of tubulin polymerization
2018 Romagnoli, Romeo; Prencipe, Filippo; Oliva, Paola; Baraldi, Stefania; Baraldi, Pier Giovanni; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Bortolozzi, Roberta; Viola, Giampietro
Synthesis, structure-activity relationships and biological evaluation of 7-phenyl-pyrroloquinolinone 3-amide derivatives as potent antimitotic agents
2017 Carta, Davide; Bortolozzi, Roberta; Sturlese, Mattia; Salmaso, Veronica; Hamel, Ernest; Basso, Giuseppe; Calderan, Laura; Quintieri, Luigi; Moro, Stefano; Viola, Giampietro; Ferlin, MARIA GRAZIA
Glucocorticoid resistance is reverted by LCK inhibition in pediatric T-cell acute lymphoblastic leukemia
2017 Serafin, Valentina; Capuzzo, Giorgia; Milani, Gloria; Minuzzo, Sonia Anna; Pinazza, Marica; Bortolozzi, Roberta; Bresolin, Silvia; Porcù, Elena; Frasson, Chiara; Indraccolo, Stefano; Basso, Giuseppe; Accordi, Benedetta
Derivati fenil-pirrolochinolinonici e loro uso
2017 Ferlin, MARIA GRAZIA; Basso, Giuseppe; Viola, Giampietro; Bortolozzi, Roberta; Carta, Davide; Moro, Stefano
Design, synthesis and biological evaluation of 3-substituted-2-oxindole hybrid derivatives as novel anticancer agents
2017 Romagnoli, Romeo; Baraldi, Pier Giovanni; Prencipe, Filippo; Oliva, Paola; Baraldi, Stefania; Salvador, Maria Kimatrai; Lopez-Cara, Luisa Carlota; Bortolozzi, Roberta; Mattiuzzo, Elena; Basso, Giuseppe; Viola, Giampietro
Synthesis and Biological Evaluation of 2-Methyl-4,5-Disubstituted Oxazoles as a Novel Class of Highly Potent Antitubulin Agents
2017 Romagnoli, Romeo; Baraldi, Pier Giovanni; Prencipe, Filippo; Oliva, Paola; Baraldi, Stefania; Salvador, Maria Kimatrai; Lopez-Cara, Luisa Carlota; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Ronca, Roberto; Bortolozzi, Roberta; Mariotto, Elena; Porcã¹, Elena; Basso, Giuseppe; Viola, Giampietro
Design and synthesis of potent in vitro and in vivo anticancer agents based on 1-(3',4',5'-trimethoxyphenyl)-2-Aryl-1H-imidazole
2016 Romagnoli, Romeo; Baraldi, Pier Giovanni; Prencipe, Filippo; Oliva, Paola; Baraldi, Stefania; Tabrizi, Mojgan Aghazadeh; Lopez-Cara, Luisa Carlota; Ferla, Salvatore; Brancale, Andrea; Hamel, Ernest; Ronca, Roberto; Bortolozzi, Roberta; Mariotto, Elena; Basso, Giuseppe; Viola, Giampietro
Design, synthesis, crystallization and biological evaluation of new symmetrical biscationic compounds as selective inhibitors of human Choline Kinase α1 (ChoKα1)
2016 Schiaffino-Ortega, Santiago; Baglioni, Eleonora; Mariotto, Elena; Bortolozzi, Roberta; Serrán-Aguilera, Luciá; Riós-Marco, Pablo; Carrasco-Jimenez, M. Paz; Gallo, Miguel A.; Hurtado-Guerrero, Ramon; Marco, Carmen; Basso, Giuseppe; Viola, Giampietro; Entrena, Antonio; López-Cara, Luisa Carlota
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