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Titolo Data di pubblicazione Autori Rivista Serie Titolo libro
Preliminary Discovery of Small Molecule Inhibitors of Epidermal Growth Factor Receptor (EGFR) That Bind to the Extracellular Domain 2022 Di Liddo, RosaVerona, MarcoVaccarin, ChristianAcquasaliente, LauraSchrenk, SandraPiccione, MonicaCenzi, CarolaDe Franco, MicheleRibaudo, GiovanniFerlin, Maria GraziaConconi, Maria TeresaChilin, AdrianaGandin, ValentinaMarzaro, Giovanni + CANCERS - -
A Novel Aza-Derivative Inhibits agr Quorum Sensing Signaling and Synergizes Methicillin-Resistant Staphylococcus aureus to Clindamycin 2021 Pauletto A.Marzaro G.Saluzzo F.Artusi I.De Filippis V.Ferlin M. G.Brun P.Castagliuolo I. + FRONTIERS IN MICROBIOLOGY - -
Multifunctional, CD44v6-targeted ORMOSIL nanoparticles enhance drugs toxicity in cancer cells 2020 Morillas-Becerril L.Peta E.Gabrielli L.Russo V.Lubian E.Ferlin M. G.Scrimin P.Palu G.Barzon L.Castagliuolo I.Mancin F.Trevisan M. + NANOMATERIALS - -
Scaffold Repurposing of in-House Chemical Library toward the Identification of New Casein Kinase 1 δinhibitors 2020 Bolcato G.Bissaro M.Valentini A.Ferlin M. G.Sturlese M.Moro S. + ACS MEDICINAL CHEMISTRY LETTERS - -
Pyridinecarboxylic acid derivative stimulates pro-angiogenic mediators by PI3K/AKT/mTOR and inhibits reactive nitrogen and oxygen species and NF-κB activation through PPARγ-dependent pathway in T. cruzi-infected macrophages 2020 Maria G. Ferlin + FRONTIERS IN IMMUNOLOGY - -
Relationship between solid state structure and solution stability of copper(ii)-hydroxypyridinecarboxylate complexes 2019 Ferlin M. G.Dean A.Di Marco V. + NEW JOURNAL OF CHEMISTRY - -
Evaluating the effects of fluorine on biological properties and metabolic stability of some antitubulin 3-substituted 7-phenyl-pyrroloquinolinones 2019 Bortolozzi R.Carta D.Dal Pra M.Mattiuzzo E.Sturlese M.Di Paolo V.Calderan L.Moro S.Quintieri L.Viola G.Ferlin M. G. + EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - -
Amidic Coupling in the Synthesis of Pyrroloquinoline 4- and 9-Carboxamides as Potential STAT3 Inhibitors 2018 Carta, DavideDal Prà, MatteoGrazia Ferlin, Maria CHEMISTRYSELECT - -
4-Hydroxy-3,5-pyridinedicarboxylic acids: synthesis, complexation properties towards Fe(III), Al(III), Cu(II), Zn(II), human serum albumin, and cellular toxicity 2018 Dean, AnnalisaFerlin, Maria GraziaParrasia, SofiaMarton, DanieleDi Marco, Valerio B. + JOURNAL OF SOLUTION CHEMISTRY - -
Synthesis and preliminary anti-inflammatory and anti-bacterial evaluation of some diflunisal aza-analogs 2018 Carta, DavideBrun, PaolaDAL PRA', MATTEOBERNABE', GIULIACastagliuolo, IgnazioFerlin, Maria Grazia MEDCHEMCOMM - -
Targeting tubulin polymerization by novel 7-aryl-pyrroloquinolinones: Synthesis, biological activity and SARs 2018 Bortolozzi, RobertaMattiuzzo, ElenaDal Pra, MatteoSturlese, MattiaMoro, StefanoCarta, DavideViola, GiampietroFerlin, Maria Grazia + EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - -
Targeting RORs nuclear receptors by novel synthetic steroidal inverse agonists for autoimmune disorders 2018 DAL PRA', MATTEOCarta, DavideSzabadkai, GyorgySuman, MatteoFrión-Herrera, YahimaPaccagnella, NicolaCastellani, GiuliaDe Martin, SaraFerlin, Maria Grazia BIOORGANIC & MEDICINAL CHEMISTRY - -
Treatment with a new peroxisome proliferator-activated receptor gamma agonist, pyridinecarboxylic acid derivative, increases angiogenesis and reduces inflammatory mediators in the heart of Trypanosoma cruzi-infected mice 2017 Carta, DavideFerlin, Maria Grazia + FRONTIERS IN IMMUNOLOGY - -
Synthesis, structure-activity relationships and biological evaluation of 7-phenyl-pyrroloquinolinone 3-amide derivatives as potent antimitotic agents 2017 CARTA, DAVIDEBORTOLOZZI, ROBERTASTURLESE, MATTIASALMASO, VERONICABASSO, GIUSEPPECALDERAN, LAURAQUINTIERI, LUIGIMORO, STEFANOVIOLA, GIAMPIETROFERLIN, MARIA GRAZIA + EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - -
Derivati fenil-pirrolochinolinonici e loro uso 2017 FERLIN, MARIA GRAZIABASSO, GIUSEPPEVIOLA, GIAMPIETROBORTOLOZZI, ROBERTACARTA, DAVIDEMORO, STEFANO - - -
The tubulin inhibitor MG-2477 induces autophagy-regulated cell death, ROS accumulation and activation of FOXO3 in neuroblastoma 2017 VIOLA, GIAMPIETROFERLIN, MARIA GRAZIA + ONCOTARGET - -
Mesoporous silica sub-micron spheres as drug dissolution enhancers: Influence of drug and matrix chemistry on functionality and stability 2016 BRIGO, LAURACAPURSO, GIOVANNIFERLIN, MARIA GRAZIABELLO, VALENTINAREALDON, NICOLABRUSATIN, GIOVANNAMORPURGO, MARGHERITA + MATERIALS SCIENCE AND ENGINEERING. C, BIOMIMETIC MATERIALS, SENSORS AND SYSTEMS - -
Synthesis of new pyrrolo-, and pyrido-anellated quinazolinones as potential antiproliferative agents 2016 CARTA, DAVIDEDALLA VIA, LISAGARCIA ARGAEZ, AIDA NELLYFERLIN, MARIA GRAZIA TETRAHEDRON - -
Novel 3-Substituted 7-Phenylpyrrolo[3,2-f]quinolin-9(6H)-ones as Single Entities with Multitarget Antiproliferative Activity 2015 CARTA, DAVIDEBORTOLOZZI, ROBERTABASSO, GIUSEPPEMORO, STEFANOVIOLA, GIAMPIETROFERLIN, MARIA GRAZIA + JOURNAL OF MEDICINAL CHEMISTRY - -
Evaluation of novel 1,3-diketone curcumin analogues and glycogen synthase kinase-3 betainhibitors as potential anti-inflammatory agents in glial cultures 2015 CARTA, DAVIDEVIOLA, GIAMPIETROMORO, STEFANOFERLIN, MARIA GRAZIA - - XXIII National Meeting in Medicinal Chemistry, Salerno, September 6-9, 2015
Mostrati risultati da 1 a 20 di 105
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