Sfoglia per Autore
Exploring the Antitumor Potential of Copper Complexes Based on Ester Derivatives of Bis(pyrazol-1-yl)acetate Ligands
2022 Pellei, Maura; Santini, Carlo; Bagnarelli, Luca; Battocchio, Chiara; Iucci, Giovanna; Venditti, Iole; Meneghini, Carlo; Amatori, Simone; Sgarbossa, Paolo; Marzano, Cristina; De Franco, Michele; Gandin, Valentina
Improvement of Kiteplatin Efficacy by a Benzoato Pt(IV) Prodrug Suitable for Oral Administration
2022 Barbanente, Alessandra; Gandin, Valentina; Ceresa, Cecilia; Marzano, Cristina; Ditaranto, Nicoletta; Hoeschele, James D; Natile, Giovanni; Arnesano, Fabio; Pacifico, Concetta; Intini, Francesco P; Margiotta, Nicola
Insight on pyrimido[5,4-g]indolizine and pyrimido[4,5-c]pyrrolo[1,2-a]azepine systems as promising photosensitizers on malignant cells
2022 Barreca, M; Ingarra, Am; Raimondi, Mv; Spanò, V; De Franco, M; Menilli, L; Gandin, V; Miolo, G; Barraja, P; Montalbano, A.
Easily Available, Amphiphilic Diiron Cyclopentadienyl Complexes Exhibit in Vitro Anticancer Activity in 2D and 3D Human Cancer Cells through Redox Modulation Triggered by CO Release
2021 Biancalana, L.; De Franco, M.; Ciancaleoni, G.; Zacchini, S.; Pampaloni, G.; Gandin, V.; Marchetti, F.
Tyrosine kinase inhibitor prodrug-loaded liposomes for controlled release at tumor microenvironment
2021 Salmaso, S.; Mastrotto, F.; Roverso, M.; Gandin, V.; De Martin, S.; Gabbia, D.; De Franco, M.; Vaccarin, C.; Verona, M.; Chilin, A.; Caliceti, P.; Bogialli, S.; Marzaro, G.
Appended Aromatic Moieties in Flexible Bis‐3‐chloropiperidines Confer Tropism against Pancreatic Cancer Cells
2021 Carraro, Caterina; Helbing, Tim; Francke, Alexander; Zuravka, Ivonne; Sosic, Alice; De Franco, Michele; Gandin, Valentina; Gatto, Barbara; Göttlich, D. Richard
Effect of chirality on the anticancer activity of Pt(ii) and Pt(iv) complexes containing 1R,2Rand 1S,2Senantiomers of thetrans-1,2-diamino-4-cyclohexene ligand (DACHEX), an analogue of diaminocyclohexane used in oxaliplatin
2021 Papadia, P.; Barbanente, A.; Ditaranto, N.; Hoeschele, J. D.; Natile, G.; Marzano, C.; Gandin, V.; Margiotta, N.
Are Pt(IV) Prodrugs That Release Combretastatin A4 True Multi-action Prodrugs?
2021 Schmidt, C.; Babu, T.; Kostrhunova, H.; Timm, A.; Basu, U.; Ott, I.; Gandin, V.; Brabec, V.; Gibson, D.
Pt(iv) complexes based on cyclohexanediamines and the histone deacetylase inhibitor 2-(2-propynyl)octanoic acid: synthesis, characterization, cell penetration properties and antitumor activity
2021 Gabano, E.; Rangone, B.; Perin, E.; Caron, G.; Ermondi, G.; Vallaro, M.; Gandin, V.; Marzano, C.; Barbanente, A.; Margiotta, N.; Ravera, M.
[99mTc(N)(DASD)(PNPn)]+ Compounds as Myocardial Perfusion Imaging Agents.
2020 Bolzati, C; Melendez-Alafort, L; Carpanese, D; De Nardo, L; Gandin, V; Marzano, C; Salvarese, N
Aromatic Linkers Unleash the Antiproliferative Potential of 3-Chloropiperidines Against Pancreatic Cancer Cells
2020 Helbing, Tim; Carraro, Caterina; Francke, Alexander; Sosic, Alice; De Franco, Michele; Gandin, Valentina; Göttlich, Richard; Gatto, Barbara
Antiproliferative Homoleptic and Heteroleptic Phosphino Silver(I) Complexes: Effect of Ligand Combination on Their Biological Mechanism of Action
2020 Dammak, K.; Porchia, M.; De Franco, M.; Zancato, M.; Naili, H.; Gandin, V.; Marzano, C.
In vitro and in vivo anticancer activity of tridentate thiosemicarbazone copper complexes: Unravelling an unexplored pharmacological target
2020 Carcelli, Mauro; Tegoni, Matteo; Bartoli, Jennifer; Marzano, Cristina; Pelosi, Giorgio; Salvalaio, Marika; Rogolino, Dominga; Gandin, Valentina
Platinum(IV) Complexes of trans-1,2-diamino-4-cyclohexene: Prodrugs Affording an Oxaliplatin Analogue that Overcomes Cancer Resistance
2020 Papadia, Paride; Micoli, Katia; Barbanente, Alessandra; Ditaranto, Nicoletta; Hoeschele, James D.; Natile, Giovanni; Marzano, Cristina; Gandin, Valentina; Margiotta, Nicola
Synthesis, characterization and biological activity of novel Cu(II) complexes of 6-methyl-2-oxo-1,2-dihydroquinoline-3-carbaldehy de-4N-substituted thiosemicarbazones
2020 Eswaran, Ramachandran; Gandin, V.; Bertani, R.; Sgarbossa, P.; Natarajan, K.; Bhuvanesh, N. S. P.; Venzo, A.; Zoleo, A.; Mozzon, M.; Dolmella, A.; Albinati, A.; Castellano, C.; Conceicao, N. R.; Guedes Da Silva, M. F. C.; Marzano, C.
In vitro antitumor activity of water-soluble copper(I) complexes with diimine and monodentate phosphine ligands
2020 Porchia, Marina; Tisato, Francesco; Zancato, Mirella; Gandin, Valentina; Marzano, Cristina
Anticancer activity, DNA binding and cell mechanistic studies of estrogen-functionalised Cu(II) complexes
2020 Barrett, S.; De Franco, M.; Kellett, A.; Dempsey, E.; Marzano, C.; Erxleben, A.; Gandin, V.; Montagner, D.
Synthesis and cytotoxic activity evaluation of new Cu(I) complexes of bis(pyrazol-1-yl) acetate ligands functionalized with an NMDA receptor antagonist
2020 Pellei, M.; Bagnarelli, L.; Luciani, L.; Del Bello, F.; Giorgioni, G.; Piergentili, A.; Quaglia, W.; De Franco, M.; Gandin, V.; Marzano, C.; Santini, C.
99mTc(N)(DASD)(pnpn)]+ (DASD=1,4-dioxa-8-azaspiro[4,5]decandithiocarba pnpn=bisphosphinoamine) for myocardial imaging
2019 Bolzati, Cristina; Salvarese, Nicola; DE NARDO, Laura; MELENDEZ ALAFORT, Laura; Gandin, Valentina; Carta, Davide; Marzano, Cristina
Expanding the Arsenal of PtIV Anticancer Agents: Multi-action PtIV Anticancer Agents with Bioactive Ligands Possessing a Hydroxy Functional Group
2019 Yempala, T.; Babu, T.; Karmakar, S.; Nemirovski, A.; Ishan, M.; Gandin, V.; Gibson, D.
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